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DESIGN OF PROTEIN KINASE INHIBITORS USING THE NATURALLY OCCURRING ISOJACAREUBIN SCAFFOLD AS A LEAD
- At: AbuDhabi (United Arab Emirates) (2019)
- Type: Poster
- Poster code: POS-DDD-010
- By: SHOEMAKE, Claire (University of Malta, Pharmacy, Malta)
- Co-author(s): Jeanelle Caruana: Pharmacy, University of Malta, Msida, Malta
Claire Shoemake: Pharmacy, University of Malta, Msida, Malta - Abstract:
Background
Protein Kinase C (PKc) is a druggable target for the mitigation of proliferative malignant disease. Isojacareubin (ISJ) is a naturally occurring molecule that has been shown to be a high affinity PKc antagonist.Methods
X-ray crystallographic deposition 2IOE describing the holo- bisindolylmaleimide (BIM) inhibitor:PKc complex was
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Last update 2 July 2026