The design of novel lead molecules using a bioisosteric approach
- At: 2013 FIP Congress in Dublin (Ireland)
- Type: Poster
- By: AZZOPARDI, Lilian (University of Malta, Msida, Malta)
- Co-author(s): Schembri, Maria (University of Malta, Msida, Malta)
Shoemake, Claire (University of Malta, Msida, Malta)
The identification of lead molecules which can be developed into drugs with clinical utility is a challenge in contemporary rational drug design. Bioisosteric manipulation and de novo design are often resorted to in this respect. This project implemented bioisosteric modification on a selected small molecule cohort in the context of a.. The access to the whole abstract and the presentation file is available to FIP members and to congress participants of that specific congress.